Pain Medicines (Analgesics) – Information for Older Adults

Plain-language information about common pain medicines in older adults. This page is for older Canadians and their caregivers. It does not replace advice from your own health-care provider.

Pain Medicines Overview

Analgesics – Medications That Relieve Pain

Main Types Acetaminophen, NSAIDs, Opioids, Other (nerve pain medicines)
Used For Headaches, Arthritis, Injuries, Post-Surgery, Chronic Pain
Key Principle Use lowest effective dose for shortest needed time
Important Note Different pain medicines have different risks – ask your provider

1. Types of common pain medicines

Pain medicines (also called analgesics) come in several types. Each works differently and has different risks and benefits, especially in older adults.

Acetaminophen

Examples: Tylenol, Atasol

Best for: Mild to moderate pain, fever

Main concern: Liver damage if too much taken

Generally safest choice for older adults when used correctly

NSAIDs

Examples: Advil (ibuprofen), Aleve (naproxen), Aspirin

Best for: Pain with inflammation (arthritis, injuries)

Main concerns: Stomach, kidneys, heart, blood pressure

Use with caution in older adults – often limited or avoided

Opioids

Examples: Codeine, morphine, oxycodone, hydromorphone

Best for: Moderate to severe pain, often short-term

Main concerns: Drowsiness, falls, confusion, constipation, dependence

Require close supervision – significant risks in older adults

Other Pain Medicines

Examples: Gabapentin, certain antidepressants, topical creams

Best for: Nerve pain, chronic pain conditions

Main concerns: Vary by medication

May be helpful for specific types of pain

The right medicine depends on you

The best pain medicine for you depends on the type of pain, your other health conditions, and what other medications you take. Always talk to your provider about which pain medicines are safest for you.

2. Acetaminophen (Tylenol, Atasol)

Acetaminophen is often the first choice for mild to moderate pain in older adults. When used within safe limits, it is generally the safest pain medicine option.

What it helps

Headaches, muscle aches, joint pain, dental pain, fever

What it doesn't do

Doesn't reduce inflammation (swelling) like NSAIDs do

Most important safety rule: Don't take too much!

Too much acetaminophen can cause serious liver damage. The maximum for most adults is 3,000–4,000 mg per day – but your provider may recommend a lower limit, especially if you're older, have liver problems, or drink alcohol.

Hidden acetaminophen – watch out!

Many products contain acetaminophen, including:

  • Cold and flu medicines (like Tylenol Cold, NyQuil)
  • Some prescription pain medicines (like Tylenol #3, Percocet)
  • Combination products for headaches, sleep, or allergies

Always check the label! It's easy to accidentally take too much if you're using multiple products. Look for "acetaminophen" or "APAP" in the ingredients.

Regular strength

325 mg per tablet – usually 1–2 tablets every 4–6 hours

Extra strength

500 mg per tablet – usually 1–2 tablets every 6–8 hours

Keep track

Write down each dose to make sure you don't exceed the daily limit

3. NSAIDs (Advil, Aleve, Aspirin, and others)

NSAIDs (Non-Steroidal Anti-Inflammatory Drugs) can help with pain and inflammation. However, they have important risks in older adults and are often limited or avoided.

Common NSAIDs

  • Ibuprofen – Advil, Motrin
  • Naproxen – Aleve, Naprosyn
  • Aspirin (at higher pain-relief doses)
  • Prescription NSAIDs – Celebrex (celecoxib), diclofenac, meloxicam

Important risks of NSAIDs in older adults

Stomach problems

Irritation, ulcers, and bleeding – can happen without warning

Kidney damage

Can worsen kidney function, especially if already reduced

High blood pressure

Can raise blood pressure and make BP medications less effective

Fluid retention

Can worsen swelling and heart failure

Heart risks

May increase risk of heart attack or stroke with long-term use

Drug interactions

Can interact with blood thinners, BP medicines, and others

When NSAIDs might be considered:

Short-term use only (a few days) for acute pain or inflammation
Lowest effective dose for the shortest time
Sometimes with a stomach-protecting medication (like omeprazole)
When benefits clearly outweigh risks for your situation

Topical NSAIDs – a safer option?

NSAID creams or gels (like Voltaren gel/diclofenac gel) applied to the skin over a painful joint may be safer than pills for localized pain like knee or hand arthritis. Less medication gets into your system. Ask your provider if this might work for you.

4. Opioids (strong pain medicines)

Opioids are powerful pain medicines that may be needed for moderate to severe pain, but they carry significant risks, especially in older adults. They require careful supervision by a health-care provider.

Common opioids

  • Codeine – often in Tylenol #3
  • Tramadol – Ultram
  • Morphine
  • Oxycodone – Percocet (with acetaminophen), OxyNEO
  • Hydromorphone – Dilaudid
  • Fentanyl – patches for chronic pain

Serious risks of opioids in older adults

Drowsiness and confusion

Can make you very sleepy and affect thinking clearly

Falls and fractures

Significantly increases fall risk – a major concern for seniors

Breathing problems

Can slow breathing dangerously, especially at higher doses

Severe constipation

Almost always happens – can be severe if not treated

Dependence

Body can become dependent – don't stop suddenly

Nausea

Can cause nausea and vomiting, especially at first

If you take opioids:

  • Take exactly as prescribed – never take more or more often
  • Start a bowel routine right away (stool softeners, laxatives as advised)
  • Don't drive or operate machinery until you know how it affects you
  • Don't mix with alcohol or other sedating medications without asking
  • Don't stop suddenly if you've been taking them regularly – your provider will taper
  • Store safely and dispose of unused medications properly

Opioids aren't always the answer

For many types of chronic pain (like arthritis or back pain), opioids may not be the best long-term choice. Studies show they often don't work better than other options for chronic pain and come with more risks. Ask your provider about all your options.

5. Other pain medicines

For certain types of pain, especially nerve pain (neuropathic pain), different medications may be used:

Gabapentin (Neurontin) and Pregabalin (Lyrica)

Used for nerve pain from diabetes, shingles, or other causes. Can cause drowsiness and dizziness, especially in older adults. Learn more about gabapentin →

Certain Antidepressants

Some antidepressants (like duloxetine, amitriptyline, nortriptyline) help with chronic pain and nerve pain, even if you're not depressed. They work on pain pathways in the brain.

Topical Treatments

Creams, gels, or patches applied to the skin – like lidocaine patches, capsaicin cream, or NSAID gels. May be safer because less medication enters your body.

Muscle Relaxants

Sometimes used for muscle spasms, but many are not recommended for older adults due to side effects like drowsiness, confusion, and falls.

6. General safety tips for pain medicines

Lowest dose, shortest time

Use the smallest amount that helps, for only as long as needed

Keep a list

Write down all pain medicines you take – prescription AND over-the-counter

Read labels carefully

Check for hidden ingredients like acetaminophen in combination products

Tell your provider everything

Include all OTC products – they need the full picture

Don't double up

Avoid taking multiple pain medicines unless your provider approves

Be careful with alcohol

Alcohol increases risks of liver damage (acetaminophen) and bleeding (NSAIDs)

Medicines to be extra careful with in older adults

Some pain medicines are on lists of "potentially inappropriate medications for older adults" because their risks often outweigh benefits. These include:

  • Long-term NSAIDs (especially in those with kidney, heart, or stomach problems)
  • Muscle relaxants like cyclobenzaprine (Flexeril) or methocarbamol
  • Meperidine (Demerol) – an opioid rarely used anymore
  • Combination products with sedating antihistamines

Ask your provider if any of your medicines are on these lists.

7. Non-drug approaches to pain

Medications aren't the only way to manage pain. Many non-drug approaches can help, often with fewer side effects. Talk to your provider about which might work for you:

Heat and cold

Ice packs for acute injuries; heat for stiff, achy muscles and joints

Gentle movement and exercise

Staying active often helps more than resting – with guidance

Physiotherapy

A physiotherapist can teach exercises and techniques for your specific pain

Massage

Can help with muscle tension and some types of pain

Mind-body approaches

Relaxation, meditation, deep breathing, and cognitive techniques

Acupuncture

May help some people with certain types of chronic pain

TENS units

Small devices that deliver mild electrical stimulation to relieve pain

Assistive devices

Canes, braces, ergonomic tools to reduce strain on painful areas

Best approach: Combination

Often the best pain management combines medications (when needed) with non-drug approaches. This can help you use lower doses of medication while still getting good pain relief.

8. When to call your doctor, nurse practitioner, or pharmacist

(Non-urgent)

Contact your health-care provider or pharmacist if:

9. When to call 911 or go to the emergency department

Call 911 immediately if:

  • Severe stomach pain with black, tarry, or bloody stools – could be bleeding
  • Vomiting blood or material that looks like coffee grounds
  • Trouble breathing or very slow breathing after taking pain medicine
  • Extreme drowsiness – you or someone else cannot be woken up after taking opioids
  • Confusion, agitation, or hallucinations after taking pain medicine
  • Signs of severe allergic reaction – swelling of face/throat, difficulty breathing, severe rash
  • Chest pain that could be heart-related

If possible, do not drive yourself. Ask someone to call for you or call an ambulance.

Naloxone (Narcan) – life-saving for opioid overdose

If you or someone you care for takes opioids, ask your pharmacist about getting a naloxone kit. Naloxone can reverse an opioid overdose and save a life. It's available free at many pharmacies in Canada.

10. Questions to ask your doctor or nurse practitioner

You can print these questions and bring them to your next appointment:

What pain medicine is safest for me given my age and health conditions?
Are there any pain medicines I should avoid completely?
How much acetaminophen is safe for me per day?
Is it safe for me to use NSAIDs like ibuprofen or naproxen?
What non-drug options might help my pain?
How long should I take this pain medicine?
Could any of my pain medicines interact with my other medications?
Would a referral to a physiotherapist or pain specialist help me?
Should I have a naloxone kit at home?